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Found 1 of ic50 data for polymerid = 50007539
TargetP2X purinoceptor(Macaca mulatta)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM254266(US10112937, Example 158 | US10150765, Example 158 ...)
Affinity DataIC50:  7.90nMAssay Description:Antagonist activity at macaque P2X7 assessed as inhibition of BzATP-induced calcium flux preincubated for 30 mins followed by BzATP addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed